

{"id":9158,"date":"2011-08-21T09:22:28","date_gmt":"2011-08-21T09:22:28","guid":{"rendered":"http:\/\/zydq.ybx8.cn\/?p=9158"},"modified":"2011-08-21T09:22:28","modified_gmt":"2011-08-21T09:22:28","slug":"%e5%b0%8f%e5%8d%87%e9%ba%bb","status":"publish","type":"post","link":"http:\/\/zydq.1006ss.com\/?p=9158","title":{"rendered":"\u5c0f\u5347\u9ebb"},"content":{"rendered":"<p>\u3010\u62fc\u97f3\u540d\u3011Xi\u01ceo Sh\u0113n\u0261 M\u00e1<\/p>\n<p>\u3010\u522b\u540d\u3011\u91d1\u4e1d\u4e09\u4e03\u3001\u5e3d\u8fab\u4e03\u3001\u5f00\u5589\u7bad\u3001\u4e09\u9762\u5200\u3001\u8336\u4e03\u3001\u767d\u5347\u9ebb\u3001\u7c73\u5347\u9ebb\u3001\u4e07\u5e74\u6839\u3001\u62d0\u67a3\u4e03\u3001\u68c9\u82b1\u4e03\u3001\u718a\u638c\u4e03<\/p>\n<p>\u3010\u6765\u6e90\u3011<br \/>\u836f\u6750\u57fa\u6e90\uff1a\u4e3a\u6bdb\u831b\u79d1\u690d\u7269\u91d1\u9f9f\u8349\u7684\u6839\u830e\u3002<br \/>\u62c9\u4e01\u690d\u7269\u52a8\u7269\u77ff\u7269\u540d\uff1aCimicifuga acerina(Sieb.et Zucc)Tanaka[C.chinensis Koidz.]<br 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\/>\u663e\u5fae\u9274\u522b\uff0c\u6839\u830e\u6a2a\u5207\u9762\uff1a\u540e\u4e00\u76ae\u5c42\u7ec6\u80de1\u5217\uff0c\u5916\u58c1\u6728\u6813\u5316\u589e\u539a\uff0c\u6709\u7684\u5916\u5e73\u5468\u58c1\u53ca\u5782\u5468\u58c1\u53ca\u5782\u5468\u58c1\u5177\u4e73\u5934\u72b6\u589e\u539a\uff0c\u7a81\u5165\u7ec6\u8154\u3002\u76ae\u5c42\u7ec6\u80de17-23\u5217\uff1b\u6709\u65f6\u53ef\u89c1\u6839\u8ff9\u7ef4\u7ba1\u675f\u3002\u4e2d\u67f1\u9798\u7ea4\u7ef4\u675f\u4e3a15-50\u4e2a\u7ea4\u7ef4\uff0c\u7ea4\u7ef4\u591a\u89d2\u5f62\u3002\u7ef4\u7ba1\u675f\u7ea628\u4e2a\uff0c\u73af\u5217\uff0c\u5916\u97e7\u578b\u3002\u97e7\u76ae\u90e8\u7ec6\u80de\u5f84\u5411\u6392\u5217\u8f83\u6574\u9f50\uff1b\u5f62\u6210\u5c42\u73af\u660e\u663e\uff0c\u54485-8\u89d2\u5f62\uff1b\u6728\u8d28\u90e8\u5bfc\u7ba1\u591a2-7\u4e2a\u6210\u7fa4\uff0c\u76f4\u5f8423-48\u03bcm\uff0c\u5185\u4fa7\u6709\u975e\u6728\u5316\u7684\u8584\u58c1\u7ec6\u80de\u7fa4\uff0c\u5176\u95f4\u6709\u5c0f\u5bfc\u7ba1\u3002\u5c04\u7ebf\u5bbd8-27\u5217\u7ec6\u80de\u3002\u9ad3\u90e8\u5927\uff0c\u5360\u6a2a\u5207\u9762\u76841\/2\u3002\u672c\u54c1\u8584\u58c1\u7ec6\u80de\u5145\u6ee1\u6dc0\u7c89\u7c92\u3002<br \/>\u7c89\u672b\u7279\u5f81\uff1a\u9ec4\u8910\u8272\u30021.\u672c\u7ea4\u7ef4\u7565\u5448\u957f\u68ad\u5f62\uff0c\u6709\u7684\u7a0d\u5f2f\u66f2\uff0c\u672b\u7aef\u659c\u5c16\u3001\u957f\u5c16\u3001\u5177\u6307\u72b6\u51f8\u8d77\u6216\u949d\u5706\uff0c\u6709\u7684\u4e8c\u53c9\u72b6\u6216\u94a9\u72b6\uff0c\u76f4\u5f849-41\u03bcm\uff0c\u957f245-374\u03bcm\uff0c\u58c1\u539a5-10\u03bcm\uff0c\u6728\u5316\uff0c\u7eb9\u5b54\u659c\u88c2\u7f1d\u72b6\u6216\u5341\u5b57\u5f62\u3001\u4eba\u5b57\u5f62\u3002<br \/>2.\u7ea4\u7ef4\u7ec6\u957f\u6839\u5f62\uff0c\u672b\u7aef\u949d\u5706\u6216\u659c\u5c16\uff0c\u76f4\u5f8429-57\u03bcm\uff0c\u957f204-408\u03bcm\uff0c\u58c1\u539a7-14\u03bcm\uff0c\u6728\u5316\u7eb9\u5b54\u5706\u70b9\u72b6\uff0c\u5b54\u6c9f\u660e\u663e\u30023.\u5bfc\u7ba1\u4e3b\u4e3a\u5177\u7f18\u7eb9\u5b54\u5bfc\u7ba1\uff0c\u4e5f\u6709\u7f51\u7eb9\uff0c\u5f31\u70b9\u7eb9\uff0c\u87ba\u7eb9\u5bfc\u7ba1\uff0c\u76f4\u5f8426-60\u03bcm\uff0c\u6709\u7684\u542b\u9ec4\u8272\u6ccc\u7269\u30024.\u6728\u8584\u58c1\u7ec6\u80de\u957f\u5706\u5f62\u6216\u7c7b\u4e09\u89d2\u5f62\uff0c\u7eb9\u5b54\u660e\u663e\uff0c\u591a\u5448\u72ed\u7f1d\u72b6\u30025.\u540e\u751f\u76ae\u5c42\u7ec6\u80de\u9ec4\u68d5\u8272\uff0c\u8868\u9762\u89c2\u7c7b\u591a\u89d2\u5f62\uff0c\u58c1\u7a0d\u539a\u30026.\u6dc0\u7c89\u7c92\u591a\u805a\u96c6\u6210\u56e2\uff0c\u5355\u7c92\u7c7b\u5706\u5f62\uff0c\u76f4\u5f843-19\u03bcm\uff1b\u590d\u7c92\u75312-3\u5206\u7c92\u7ec4\u6210\u3002<\/p>\n<p>\u3010\u5316\u5b66\u6210\u4efd\u3011\u6839\u830e\u542b\u4ee5\u5347\u9ebb\u73af\u6c27\u9187(cimigenol)\uff0c25-O-\u7532\u57fa\u5347\u9ebb\u73af\u6c27\u9187\uff0c15-O-\u7532\u57fa\u5347\u9ebb\u73af\u6c27\u9187\uff0c\u53bb\u7f9f-15-O-\u7532\u57fa\u5347\u9ebb\u73af\u6c27\u9187\uff0c25-O-\u4e59\u9170\u5347\u9ebb\u73af\u6c27\u9187\uff0c15\uff0c24-\u53cc\u5f02\u5347\u73af\u6c27\u9187(cimigol)\uff0c\u5174\u5b89\u5347\u9ebb\u9187(dahurinol)\uff0c\u5f02\u5174\u5b89\u5347\u9ebb\u9187(isodahurinol)\uff0c25-O-\u7532\u57fa\u5f02\u5174\u5b89\u5347\u9ebb\u9187\uff0c\u91d1\u9f9f\u8349\u4e8c\u9187(acerinol)\uff0c25-O-\u7532\u57fa\u91d1\u9f9f\u8349\u4e8c\u9187\uff0c\u91d1\u7535\u916e\u9187(acerionol)\uff0c24-O-\u4e59\u9170\u91d1\u7535\u8349\u916e\u9187\uff0cO-\u7532\u57fa\u91d1\u9f9f\u8349\u9187(O-methylcimiacerol)\u7b49\u4e3a\u7519\u5143\u7684\u7cd6\u7519\uff1b\u8fd8\u542b\u6709\u03b2-\u8c37\u753e\u9187(\u03b2-sitosterol),15,24-\u4ee5\u4ee5\u5f02\u5347\u9ebb\u73af\u6c27\u9187\uff0c\u5174\u5b89\u5347\u9ebb\u9187\uff0c\u5f02\u5174\u5b89\u5404\u9ebb\u9187\uff0c\u5347\u9ebb\u4e8c\u70ef\u9187(cimicifugenol)\uff0c\u5347\u9ebb\u4e8c\u7076\u70ef\u9187\u916f\uff0c25-O-\u4e59\u9170\u5347\u9ebb\u73af\u6c27\u9187\u6728\u7cae\u7519(25-o-acetylcimigenoside)\uff0c25-O-\u7532\u7519\u57fa\u5347\u9ebb\u73af\u6c27\u9187\u6728\u7cd6\u7519\uff0c\u5347\u9ebb\u7519(cimicifugoside)\uff0c\u5347\u9ebb\u65b0\u9187\u6728\u7cd6\u7519(shenfgmanolxyloside)\uff0c\u4e59\u9170\u5347\u9ebb\u65b0\u9187\u6728\u7cd6\u7519\u53ca24-\u4e59\u9170\u57fa\u6c34\u5408\u5347\u9ebb\u65b0\u9187\u6728\u7cd6\u7519(24-acetylhydrosjhengmanol xyloside)\uff0c\u5e76\u8ba4\u4e3a\u65b0\u9c9c\u91d1\u7535\u8349\u6839\u830e\u4e0d\u542b25-O-\u4e59\u9170\u53ca25-O-\u7532\u57fa\u5347\u9ebb\u73af\u6c27\u9187\u6728\u7cd6\u7519\uff0c\u5b83\u4eec\u662f\u5206\u79bb\u6210\u8fc7\u7a0b\u4e2d\u4ea7\u751f\u7684\u4eba\u5de5\u77eb\u4f5c\u7269\u3002<\/p>\n<p>\u3010\u9274\u522b\u3011\u7406\u5316\u9274\u522b\uff0c\u8584\u5c42\u8272\u8c31\uff1a\u53d6\u672c\u54c1\u7c89\u672b(40\u76ee)\u5c11\u8bb8\uff0c\u52a0\u7532\u9187\u9002\u91cf\uff0c\u51b7\u6d7848h\uff0c\u6ee4\u8fc7\u3002\u6ee4\u6db2\u6d53\u7f29\u81f3\u5e72\uff0c\u52a0\u7532\u91871ml\u6eb6\u89e3\uff0c\u4e3a\u6837\u5415\u6db2\u3002\u53e6\u4ee5\u963f\u9b4f\u9178(AR)\u3001\u5496\u5561\u9178(AR)\u52a0\u9002\u91cf\u7532\u9187\u6eb6\u89e3\u4f5c\u4e3a\u5bf9\u7167\u54c1\u6db2\u3002\u5206\u522b\u5438\u53d6\u6837\u54c1\u6db2\u548c\u5bf9\u7167\u54c1\u6db2\u54045\u03bcl\u70b9\u4e8e\u594e 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